ALEXANDRIA, Va., Sept. 17 -- United States Patent no. 12,414,952, issued on Sept. 16, was assigned to Merck Sharp & Dohme LLC (Rahway, N.J.).
"Substituted amino triazolopyrimidine and amino triazolopyrazine adenosine receptor antagonists, pharmaceutical compositions and their use" was invented by Zachary G. Brill (Boston), Amjad Ali (Freehold, N.J.), Jared Cumming (Winchester, Mass.), Duane DeMong (Hanover, Mass.), Qiaolin Deng (Edison, N.J.), Gioconda V. Gallo-Etienne (New Providence, N.J.), Thomas H. Graham (Somerville, Mass.), Rongze Kuang (Green Brook, N.J.), Matthew A. Larsen (Dedham, Mass.), Yeon-Hee Lim (South San Francisco, Calif.), Kun Liu (Needham, Mass.), Umar Faruk Mansoor (Hopkinton, Mass.), Jesus Moreno (Dorchester Center, Ma...